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Endogenous G(s)-Coupled Receptors in Smooth Muscle Exhibit Differential Susceptibility to GRK2/3-Mediated Desensitization

Although G protein-coupled receptor (GPCR) kinases (GRKs) have been shown to mediate desensitization of numerous GPCRs in studies using cellular expression systems, their function under physiological conditions is less well understood. In the current study, we employed various strategies to assess t...

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Autori principali: Kong, Kok Choi, Gandhi, Uma, Martin, T. J., Anz, Candace B., Yan, Huandong, Misior, Anna M., Pascual, Rodolfo M., Deshpande, Deepak A., Penn, Raymond B.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2008
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2947145/
https://ncbi.nlm.nih.gov/pubmed/18690720
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/bi801056w
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