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The Mibefradil Derivative NNC55-0396, a Specific T-Type Calcium Channel Antagonist, Exhibits Less CYP3A4 Inhibition than Mibefradil

A novel mibefradil derivative, NNC55-0396, designed to be hydrolysis resistant was shown to be a selective T-type Ca(2+) channel inhibitor without L-type Ca(2+) channel efficacy. However, its effects on cytochrome P450s have not previously been examined. We investigated the inhibitory effects of NNC...

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Detalhes bibliográficos
Main Authors: Bui, Peter H., Quesada, Arnulfo, Handforth, Adrian, Hankinson, Oliver
Formato: Artigo
Idioma:Inglês
Publicado em: 2008
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2927974/
https://ncbi.nlm.nih.gov/pubmed/18411403
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.107.020115
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