Načítá se...

The Mibefradil Derivative NNC55-0396, a Specific T-Type Calcium Channel Antagonist, Exhibits Less CYP3A4 Inhibition than Mibefradil

A novel mibefradil derivative, NNC55-0396, designed to be hydrolysis resistant was shown to be a selective T-type Ca(2+) channel inhibitor without L-type Ca(2+) channel efficacy. However, its effects on cytochrome P450s have not previously been examined. We investigated the inhibitory effects of NNC...

Celý popis

Uloženo v:
Podrobná bibliografie
Hlavní autoři: Bui, Peter H., Quesada, Arnulfo, Handforth, Adrian, Hankinson, Oliver
Médium: Artigo
Jazyk:Inglês
Vydáno: 2008
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC2927974/
https://ncbi.nlm.nih.gov/pubmed/18411403
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.107.020115
Tagy: Přidat tag
Žádné tagy, Buďte první, kdo otaguje tento záznam!