Loading...

Eribulin Binds at Microtubule Ends to a Single Site on Tubulin to Suppress Dynamic Instability

Eribulin mesylate (E7389), a synthetic analog of the marine natural product halichondrin B, is in Phase III clinical trials for the treatment of cancer. Eribulin targets microtubules, suppressing dynamic instability at microtubule plus ends through an inhibition of microtubule growth with little or...

Full description

Saved in:
Bibliographic Details
Main Authors: Smith, Jennifer A., Wilson, Leslie, Azarenko, Olga, Zhu, Xiaojie, Lewis, Bryan M., Littlefield, Bruce A., Jordan, Mary Ann
Format: Artigo
Language:Inglês
Published: 2010
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC2846717/
https://ncbi.nlm.nih.gov/pubmed/20030375
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/bi901810u
Tags: Add Tag
No Tags, Be the first to tag this record!