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Eribulin Binds at Microtubule Ends to a Single Site on Tubulin to Suppress Dynamic Instability

Eribulin mesylate (E7389), a synthetic analog of the marine natural product halichondrin B, is in Phase III clinical trials for the treatment of cancer. Eribulin targets microtubules, suppressing dynamic instability at microtubule plus ends through an inhibition of microtubule growth with little or...

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Autors principals: Smith, Jennifer A., Wilson, Leslie, Azarenko, Olga, Zhu, Xiaojie, Lewis, Bryan M., Littlefield, Bruce A., Jordan, Mary Ann
Format: Artigo
Idioma:Inglês
Publicat: 2010
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2846717/
https://ncbi.nlm.nih.gov/pubmed/20030375
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/bi901810u
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