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Potent inhibitors of furin and furin-like proprotein convertases containing decarboxylated P1 arginine mimetics

Furin belongs to the family of proprotein convertases (PCs) and is involved in numerous normal physiological and pathogenic processes, such as viral propagation, bacterial toxin activation, cancer and metastasis. Furin and related furin-like PCs cleave their substrates at characteristic multibasic c...

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Detalhes bibliográficos
Main Authors: Becker, Gero L., Sielaff, Frank, Than, Manuel E., Lindberg, Iris, Routhier, Sophie, Day, Robert, Lu, Yinghui, Garten, Wolfgang, Steinmetzer, Torsten
Formato: Artigo
Idioma:Inglês
Publicado em: 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2834293/
https://ncbi.nlm.nih.gov/pubmed/20038105
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm9012455
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