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Novel effects mediated by bradykinin and pharmacological characterization of bradykinin B(2) receptor antagonism in human synovial fibroblasts

BACKGROUND AND PURPOSE: Bradykinin (BK) and B(2) receptors have been implicated in the pathophysiology of osteoarthritis (OA), and synovitis is one of its hallmarks. Here, the selective B(2) receptor antagonists MEN16132 and icatibant have been pharmacologically characterized in human synovial cells...

पूर्ण विवरण

में बचाया:
ग्रंथसूची विवरण
मुख्य लेखकों: Bellucci, F, Cucchi, P, Catalani, C, Giuliani, S, Meini, S, Maggi, CA
स्वरूप: Artigo
भाषा:Inglês
प्रकाशित: Blackwell Publishing Ltd 2009
विषय:
ऑनलाइन पहुंच:https://ncbi.nlm.nih.gov/pmc/articles/PMC2807661/
https://ncbi.nlm.nih.gov/pubmed/20050188
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/j.1476-5381.2009.00511.x
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