Caricamento...

Engineering of a novel hybrid enzyme: an anti-inflammatory drug target with triple catalytic activities directly converting arachidonic acid into the inflammatory prostaglandin E(2)

Cyclooxygenase isoform-2 (COX-2) and microsomal prostaglandin E(2) synthase-1 (mPGES-1) are inducible enzymes that become up-regulated in inflammation and some cancers. It has been demonstrated that their coupling reaction of converting arachidonic acid (AA) into prostaglandin (PG) E(2) (PGE(2)) is...

Descrizione completa

Salvato in:
Dettagli Bibliografici
Autori principali: Ruan, Ke-He, Cervantes, Vanessa, So, Shui-Ping
Natura: Artigo
Lingua:Inglês
Pubblicazione: Oxford University Press 2009
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2777022/
https://ncbi.nlm.nih.gov/pubmed/19850676
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/protein/gzp058
Tags: Aggiungi Tag
Nessun Tag, puoi essere il primo ad aggiungerne! !