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Shape shifting leads to small molecule allosteric drug discovery

Enzymes that regulate their activity by modulating an equilibrium of alternate, non-additive, functionally distinct oligomeric assemblies (morpheeins) define a novel mode of allostery (Jaffe, TiBS 30:490-7, 2005). The oligomeric equilibrium for porphobilinogen synthase (PBGS) consists of high-activi...

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Bibliografiske detaljer
Main Authors: Lawrence, Sarah H., Ramirez, Ursula D., Tang, Lei, Fazliyev, Farit, Kundrat, Lenka, Markham, George D., Jaffe, Eileen K.
Format: Artigo
Sprog:Inglês
Udgivet: 2008
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC2703447/
https://ncbi.nlm.nih.gov/pubmed/18559269
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.chembiol.2008.04.012
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