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CYP2C9 Amino Acid Residues Influencing Phenytoin Turnover and Metabolite Regio- and Stereochemistry

Phenytoin has been an effective anticonvulsant agent for over 60 years, although its clinical use is complicated by nonlinear pharmacokinetics, a narrow therapeutic index, and metabolically based drug-drug interactions. Although it is well established that CYP2C9 is the major cytochrome P450 enzyme...

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Autori principali: Mosher, Carrie M., Tai, Guoying, Rettie, Allan E.
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Society for Pharmacology and Experimental Therapeutics 2009
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2683772/
https://ncbi.nlm.nih.gov/pubmed/19258521
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/jpet.109.150706
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