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Kinetic and structural studies of phosphodiesterase-8A and implication on the inhibitor selectivity

Cyclic nucleotide phosphodiesterase-8 (PDE8) is a family of cAMP-specific enzymes and plays important roles in many biological processes, including T-cell activation, testosterone production, adrenocortical hyperplasia, and thyroid function. However, no PDE8 selective inhibitors are available for tr...

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Autors principals: Wang, Huanchen, Yan, Zier, Yang, Serena, Cai, Jiwen, Robinson, Howard, Ke, Hengming
Format: Artigo
Idioma:Inglês
Publicat: 2008
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2646200/
https://ncbi.nlm.nih.gov/pubmed/18983167
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/bi801487x
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