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A Formal [3,3]-Sigmatropic Rearrangement Route to Quaternary α-Vinyl Amino Acids: Use of Allylic N-PMP Trifluoroacetimidates

Pd(II)-mediated rearrangement of allylic N-PMP (p-methoxyphenyl) trifluoroacetimidates provides the first formal sigmatropic route to quaternary, α-vinylic amino acids, potential suicide substrates for PLP-enzymes. The amino acid side chains enter via transition metal-mediated C-C bond constructions...

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Detaylı Bibliyografya
Asıl Yazarlar: Berkowitz, David B., Wu, Bin, Li, Huijie
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: 2006
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC2504469/
https://ncbi.nlm.nih.gov/pubmed/16494487
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ol060019s
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