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Application of high-throughput screening to identify a novel αIIb-specific small- molecule inhibitor of αIIbβ3-mediated platelet interaction with fibrinogen

Small-molecule αIIbβ3 antagonists competitively block ligand binding by spanning between the D224 in αIIb and the MIDAS metal ion in β3. They variably induce conformational changes in the receptor, which may have undesirable consequences. To identify αIIbβ3 antagonists with novel structures, we test...

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Main Authors: Blue, Robert, Murcia, Marta, Karan, Charles, Jiroušková, Markéta, Coller, Barry S.
格式: Artigo
語言:Inglês
出版: American Society of Hematology 2008
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在線閱讀:https://ncbi.nlm.nih.gov/pmc/articles/PMC2214768/
https://ncbi.nlm.nih.gov/pubmed/17978171
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1182/blood-2007-08-105544
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