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Synthesis and SAR of conformationally restricted inhibitors of soluble epoxide hydrolase

A series of conformationally restricted inhibitors of human soluble epoxide hydrolase (sEH) has been developed. Inhibition potency of the described compounds ranges from 4.2 μM to 1.1 nM against recombinant sEH. N-(1-Acetylpiperidin-4-yl)-N′-(adamant-1-yl) urea (5a) was found to be a potent inhibito...

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Detalhes bibliográficos
Main Authors: Jones, Paul D., Tsai, Hsing-Ju, Do, Zung N., Morisseau, Christophe, Hammock, Bruce D.
Formato: Artigo
Idioma:Inglês
Publicado em: 2006
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC1904344/
https://ncbi.nlm.nih.gov/pubmed/16870439
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2006.07.009
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