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Peptidyl-urea based inhibitors of soluble epoxide hydrolases

We prepared a series of amino acid derived cyclohexyl and adamantyl ureas and tested them as inhibitors of the human soluble epoxide hydrolase, and obtained very potent compounds (K(I) = 15 nM) that are >10-fold more soluble than previously described sEH inhibitors. While our lead compound 2 show...

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Hlavní autoři: Morisseau, Christophe, Newman, John W., Tsai, Hsing-Ju, Baecker, Preston A., Hammock, Bruce D.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2006
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC1892215/
https://ncbi.nlm.nih.gov/pubmed/16908134
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2006.07.073
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