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Novel 1-8-bridged chiral quinolones with activity against topoisomerase II: stereospecificity of the eukaryotic enzyme.

A series of novel C-7 quinolyl-substituted enantiomers of ofloxacin were used to determine the stereospecificity of topoisomerase II for the C-11 methyl group in tricyclic quinolones. In all cases, the S isomer was the most active compound against the eukaryotic enzyme. It was approximately 2.2-fold...

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Bibliographic Details
Main Authors: Froelich-Ammon, S J, McGuirk, P R, Gootz, T D, Jefson, M R, Osheroff, N
Format: Artigo
Language:Inglês
Published: 1993
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC187729/
https://ncbi.nlm.nih.gov/pubmed/8388196
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