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Increased hindrance on the chiral carbon atom of mexiletine enhances the block of rat skeletal muscle Na(+) channels in a model of myotonia induced by ATX

1. The antiarrhythmic drug mexiletine (Mex) is also used against myotonia. Searching for a more efficient drug, a new compound (Me5) was synthesized substituting the methyl group on the chiral carbon atom of Mex by an isopropyl group. Effects of Me5 on Na(+) channels were compared to those of Mex in...

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Bibliografiska uppgifter
Huvudupphovsmän: Desaphy, Jean-François, Camerino, Diana Conte, Franchini, Carlo, Lentini, Giovanni, Tortorella, Vincenzo, De Luca, Annamaria
Materialtyp: Artigo
Språk:Inglês
Publicerad: 1999
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Länkar:https://ncbi.nlm.nih.gov/pmc/articles/PMC1571747/
https://ncbi.nlm.nih.gov/pubmed/10578128
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0702901
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