AMD3100, a CxCR4 Antagonist, Attenuates Allergic Lung Inflammation and Airway Hyperreactivity

Por Lukacs, Nicholas W., Berlin, Aaron, Schols, Dominique, Skerlj, Renato T., Bridger, Gary J.
Publicado em 2002

Electrophilic Helical Peptides That Bond Covalently, Irreversibly, and Selectively in a Protein–Protein Interaction Site

Por de Araujo, Aline Dantas, Lim, Junxian, Good, Andrew C., Skerlj, Renato T., Fairlie, David P.
Publicado no ACS Med Chem Lett (2016)

The orally bioavailable allosteric CXCR4 HIV-1 entry inhibitor AMD11070

Por Fricker, Simon, Mosi, Renee, Anastassova, Virginia, Labrecque, Jean, Wong, Rebecca, Skerlj, Renato, Bridger, Gary, Huskens, Dana, Schols, Dominique
Publicado em 2012

Inhibition of Human Immunodeficiency Virus Replication by a Dual CCR5/CXCR4 Antagonist

Por Princen, Katrien, Hatse, Sigrid, Vermeire, Kurt, Aquaro, Stefano, De Clercq, Erik, Gerlach, Lars-Ole, Rosenkilde, Mette, Schwartz, Thue W., Skerlj, Renato, Bridger, Gary, Schols, Dominique
Publicado em 2004

Optimization of Potent Inhibitors of P. falciparum Dihydroorotate Dehydrogenase for the Treatment of Malaria

Por Skerlj, Renato T., Bastos, Cecilia M., Booker, Michael L., Kramer, Martin L., Barker, Robert H., Celatka, Cassandra A., O’Shea, Thomas J., Munoz, Benito, Sidhu, Amar Bir, Cortese, Joseph F., Wittlin, Sergio, Papastogiannidis, Petros, Angulo-Barturen, Inigo, Jimenez-Diaz, Maria Belen, Sybertz, Edmund
Publicado em 2011

Mitigating hERG Inhibition: Design of Orally Bioavailable CCR5 Antagonists as Potent Inhibitors of R5 HIV-1 Replication

Por Skerlj, Renato, Bridger, Gary, Zhou, Yuanxi, Bourque, Elyse, McEachern, Ernest, Danthi, Sanjay, Langille, Jonathan, Harwig, Curtis, Veale, Duane, Carpenter, Bryon, Ba, Tuya, Bey, Michael, Baird, Ian, Wilson, Trevor, Metz, Markus, MacFarland, Ron, Mosi, Renee, Bodart, Veronique, Wong, Rebecca, Fricker, Simon, Huskens, Dana, Schols, Dominique
Publicado em 2012

Novel Inhibitors of Plasmodium falciparum Dihydroorotate Dehydrogenase with Anti-malarial Activity in the Mouse Model

Por Booker, Michael L., Bastos, Cecilia M., Kramer, Martin L., Barker, Robert H., Skerlj, Renato, Sidhu, Amar Bir, Deng, Xiaoyi, Celatka, Cassandra, Cortese, Joseph F., Guerrero Bravo, Jose E., Crespo Llado, Keila N., Serrano, Adelfa E., Angulo-Barturen, Iñigo, Jiménez-Díaz, María Belén, Viera, Sara, Garuti, Helen, Wittlin, Sergio, Papastogiannidis, Petros, Lin, Jing-wen, Janse, Chris J., Khan, Shahid M., Duraisingh, Manoj, Coleman, Bradley, Goldsmith, Elizabeth J., Phillips, Margaret A., Munoz, Benito, Wirth, Dyann F., Klinger, Jeffrey D., Wiegand, Roger, Sybertz, Edmund
Publicado em 2010

Aminoindoles, a Novel Scaffold with Potent Activity against Plasmodium falciparum

Por Barker, Robert H., Urgaonkar, Sameer, Mazitschek, Ralph, Celatka, Cassandra, Skerlj, Renato, Cortese, Joseph F., Tyndall, Erin, Liu, Hanlan, Cromwell, Mandy, Sidhu, Amar Bir, Guerrero-Bravo, Jose E., Crespo-Llado, Keila N., Serrano, Adelfa E., Lin, Jing-wen, Janse, Chris J., Khan, Shahid M., Duraisingh, Manoj, Coleman, Bradley I., Angulo-Barturen, Inigo, Jiménez-Díaz, María Belén, Magán, Noemí, Gomez, Vanesa, Ferrer, Santiago, Martínez, María Santos, Wittlin, Sergio, Papastogiannidis, Petros, O'Shea, Thomas, Klinger, Jeffrey D., Bree, Mark, Lee, Edward, Levine, Mikaela, Wiegand, Roger C., Munoz, Benito, Wirth, Dyann F., Clardy, Jon, Bathurst, Ian, Sybertz, Edmund
Publicado em 2011