Bioluminescence Resonance Energy Transfer Based G Protein-Activation Assay to Probe Duration of Antagonism at the Histamine H(3) Receptor

Tekijä Mocking, Tamara A. M., Buzink, Maurice C. M. L., Leurs, Rob, Vischer, Henry F.
Julkaisussa Int J Mol Sci (2019)

A Photoswitchable Agonist for the Histamine H(3) Receptor, a Prototypic Family A G‐Protein‐Coupled Receptor

Tekijä Hauwert, Niels J., Mocking, Tamara A. M., Da Costa Pereira, Daniel, Lion, Ken, Huppelschoten, Yara, Vischer, Henry F., De Esch, Iwan J. P., Wijtmans, Maikel, Leurs, Rob
Julkaisussa Angew Chem Int Ed Engl (2019)

Covalent Inhibition of the Histamine H(3) Receptor

Tekijä Wágner, Gábor, Mocking, Tamara A. M., Kooistra, Albert J., Slynko, Inna, Ábrányi-Balogh, Péter, Keserű, György M., Wijtmans, Maikel, Vischer, Henry F., de Esch, Iwan J. P., Leurs, Rob
Julkaisussa Molecules (2019)

A toolbox of molecular photoswitches to modulate the CXCR3 chemokine receptor with light

Tekijä Gómez-Santacana, Xavier, de Munnik, Sabrina M, Mocking, Tamara A M, Hauwert, Niels J, Sun, Shanliang, Vijayachandran, Prashanna, de Esch, Iwan J P, Vischer, Henry F, Wijtmans, Maikel, Leurs, Rob
Julkaisussa Beilstein J Org Chem (2019)

4-(3-Aminoazetidin-1-yl)pyrimidin-2-amines as High-Affinity Non-imidazole Histamine H(3) Receptor Agonists with in Vivo Central Nervous System Activity

Tekijä Wágner, Gábor, Mocking, Tamara A. M., Arimont, Marta, Provensi, Gustavo, Rani, Barbara, Silva-Marques, Bruna, Latacz, Gniewomir, Da Costa Pereira, Daniel, Karatzidou, Christina, Vischer, Henry F., Wijtmans, Maikel, Kieć-Kononowicz, Katarzyna, de Esch, Iwan J. P., Leurs, Rob
Julkaisussa J Med Chem (2019)

Synthesis and Characterization of a Bidirectional Photoswitchable Antagonist Toolbox for Real-Time GPCR Photopharmacology

Tekijä Hauwert, Niels J., Mocking, Tamara A. M., Da Costa Pereira, Daniel, Kooistra, Albert J., Wijnen, Lisa M., Vreeker, Gerda C. M., Verweij, Eléonore W. E., De Boer, Albertus H., Smit, Martine J., De Graaf, Chris, Vischer, Henry F., de Esch, Iwan J. P., Wijtmans, Maikel, Leurs, Rob
Julkaisussa J Am Chem Soc (2018)