Active site and allosteric inhibitors of the ribonuclease H activity of HIV reverse transcriptase

od Corona, Angela, Masaoka, Takashi, Tocco, Graziella, Tramontano, Enzo, Le Grice, Stuart FJ
Izdano u Future Med Chem (2013)

A cell-free enzymatic activity assay for the evaluation of HIV-1 drug resistance to protease inhibitors

od Matsunaga, Satoko, Masaoka, Takashi, Sawasaki, Tatsuya, Morishita, Ryo, Iwatani, Yasumasa, Tatsumi, Masashi, Endo, Yaeta, Yamamoto, Naoki, Sugiura, Wataru, Ryo, Akihide
Izdano u Front Microbiol (2015)

Traceless Solid-Phase α-Hydroxytropolone Synthesis

od D’Erasmo, Michael P., Masaoka, Takashi, Wilson, Jennifer A., Hunte, Errol M., Beutler, John A., Le Grice, Stuart F. J., Murelli, Ryan P.
Izdano u Medchemcomm (2016)

Exploiting Drug-Resistant Enzymes as Tools to Identify Thienopyrimidinone Inhibitors of Human Immunodeficiency Virus Reverse Transcriptase-Associated Ribonuclease H

od Masaoka, Takashi, Chung, Suhman, Caboni, Pierluigi, Rausch, Jason W., Wilson, Jennifer A., Taskent-Sezgin, Humeyra, Beutler, John A., Tocco, Graziella, Le Grice, Stuart F. J.
Izdano 2013

Ribonuclease H/DNA Polymerase HIV-1 Reverse Transcriptase Dual Inhibitor: Mechanistic Studies on the Allosteric Mode of Action of Isatin-Based Compound RMNC6

od Corona, Angela, Meleddu, Rita, Esposito, Francesca, Distinto, Simona, Bianco, Giulia, Masaoka, Takashi, Maccioni, Elias, Menéndez-Arias, Luis, Alcaro, Stefano, Le Grice, Stuart F. J., Tramontano, Enzo
Izdano u PLoS One (2016)

Sesquiterpenoid Tropolone Glycosides from Liriosma ovata

od Ma, Jun, Pawar, Rahul S., Grundel, Erich, Mazzola, Eugene P., Ridge, Clark D., Masaoka, Takashi, Le Grice, Stuart F. J., Wilson, Jennifer, Beutler, John A., Krynitsky, Alexander J.
Izdano u J Nat Prod (2015)

Unique Flap Conformation in an HIV-1 Protease with High-Level Darunavir Resistance

od Nakashima, Masaaki, Ode, Hirotaka, Suzuki, Koji, Fujino, Masayuki, Maejima, Masami, Kimura, Yuki, Masaoka, Takashi, Hattori, Junko, Matsuda, Masakazu, Hachiya, Atsuko, Yokomaku, Yoshiyuki, Suzuki, Atsuo, Watanabe, Nobuhisa, Sugiura, Wataru, Iwatani, Yasumasa
Izdano u Front Microbiol (2016)

Studies on Cycloheptathiophene-3-Carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H inhibitors

od Corona, Angela, Desantis, Jenny, Massari, Serena, Distinto, Simona, Masaoka, Takashi, Sabatini, Stefano, Esposito, Francesca, Manfroni, Giuseppe, Maccioni, Elias, Cecchetti, Violetta, Pannecouque, Christophe, Le Grice, Stuart F.J., Tramontano, Enzo, Tabarrini, Oriana
Izdano u ChemMedChem (2016)

Synthetic α-Hydroxytropolones as Inhibitors of HIV Reverse Transcriptase Ribonuclease H Activity()

od Murelli, Ryan P., D'Erasmo, Michael P., Hirsch, Danielle R., Meck, Christine, Masaoka, Takashi, Wilson, Jennifer A., Zhang, Baofeng, Pal, Rajat K., Gallicchio, Emilio, Beutler, John A., Le Grice, Stuart F. J.
Izdano u Medchemcomm (2016)

Characterization of the C-Terminal Nuclease Domain of Herpes Simplex Virus pUL15 as a Target of Nucleotidyltransferase Inhibitors

od Masaoka, Takashi, Zhao, Haiyan, Hirsch, Danielle R., D'Erasmo, Michael P., Meck, Christine, Varnado, Brittany, Gupta, Ankit, Meyers, Marvin J., Baines, Joel, Beutler, John A., Murelli, Ryan P., Tang, Liang, Le Grice, Stuart F. J.
Izdano u Biochemistry (2016)

Lack of Association between Intact/Deletion Polymorphisms of the APOBEC3B Gene and HIV-1 Risk

od Imahashi, Mayumi, Izumi, Taisuke, Watanabe, Dai, Imamura, Junji, Matsuoka, Kazuhiro, Ode, Hirotaka, Masaoka, Takashi, Sato, Kei, Kaneko, Noriyo, Ichikawa, Seiichi, Koyanagi, Yoshio, Takaori-Kondo, Akifumi, Utsumi, Makoto, Yokomaku, Yoshiyuki, Shirasaka, Takuma, Sugiura, Wataru, Iwatani, Yasumasa, Naoe, Tomoki
Izdano 2014

Sensitivity of the C-Terminal Nuclease Domain of Kaposi's Sarcoma-Associated Herpesvirus ORF29 to Two Classes of Active-Site Ligands

od Miller, Jennifer T., Zhao, Haiyan, Masaoka, Takashi, Varnado, Brittany, Cornejo Castro, Elena M., Marshall, Vickie A., Kouhestani, Kaivon, Lynn, Anna Y., Aron, Keith E., Xia, Anqi, Beutler, John A., Hirsch, Danielle R., Tang, Liang, Whitby, Denise, Murelli, Ryan P., Le Grice, Stuart F. J.
Izdano u Antimicrob Agents Chemother (2018)