Structure-Activity Relationships of Constrained Phenylethylamine Ligands for the Serotonin 5-HT(2) Receptors

Por Isberg, Vignir, Paine, James, Leth-Petersen, Sebastian, Kristensen, Jesper L., Gloriam, David E.
Publicado em 2013

Correction: Structure-Activity Relationships of Constrained Phenylethylamine Ligands for the Serotonin 5-HT(2) Receptors

Por Isberg, Vignir, Paine, James, Leth-Petersen, Sebastian, Kristensen, Jesper L., Gloriam, David E.
Publicado em 2014

Crystal Structure of Lymnaea stagnalis AChBP Complexed with the Potent nAChR Antagonist DHβE Suggests a Unique Mode of Antagonism

Por Shahsavar, Azadeh, Kastrup, Jette S., Nielsen, Elsebet Ø., Kristensen, Jesper L., Gajhede, Michael, Balle, Thomas
Publicado em 2012

Hallucinogen-like effects of 2-([2-(4-cyano-2,5-dimethoxyphenyl) ethylamino]methyl)phenol (25CN-NBOH), a novel N-benzylphenethylamine with 100-fold selectivity for 5-HT(2A) recepto...

Por Fantegrossi, William E., Gray, Bradley W., Bailey, Jessica M., Smith, Douglas, Hansen, Martin, Kristensen, Jesper L.
Publicado no Psychopharmacology (Berl) (2014)

Synthesis and Structure–Activity Relationships of N-Benzyl Phenethylamines as 5-HT(2A/2C) Agonists

Por Hansen, Martin, Phonekeo, Karina, Paine, James S., Leth-Petersen, Sebastian, Begtrup, Mikael, Bräuner-Osborne, Hans, Kristensen, Jesper L.
Publicado em 2014

Dissecting the Binding Mode of Low Affinity Phage Display Peptide Ligands to Protein Targets by Hydrogen/Deuterium Exchange Coupled to Mass Spectrometry

Por Leurs, Ulrike, Lohse, Brian, Ming, Shonoi, Cole, Philip A., Clausen, Rasmus P., Kristensen, Jesper L., Rand, Kasper D.
Publicado no Anal Chem (2014)

Synthesis and In Vitro Evaluation of Oxindole Derivatives as Potential Radioligands for 5-HT(7) Receptor Imaging with PET

Por Herth, Matthias M., Volk, Balázs, Pallagi, Katalin, Kofoed Bech, Lasse, Antoni, Ferenc A., Knudsen, Gitte M., Kristensen, Jesper L.
Publicado em 2012

Posttranslational Modifications of the Histone 3 Tail and Their Impact on the Activity of Histone Lysine Demethylases In Vitro

Por Lohse, Brian, Helgstrand, Charlotte, Kristensen, Jan B. L., Leurs, Ulrike, Cloos, Paul A. C., Kristensen, Jesper L., Clausen, Rasmus P.
Publicado em 2013

Substrate- and Cofactor-independent Inhibition of Histone Demethylase KDM4C

Por Leurs, Ulrike, Lohse, Brian, Rand, Kasper D., Ming, Shonoi, Riise, Erik S., Cole, Philip A., Kristensen, Jesper L., Clausen, Rasmus P.
Publicado em 2014

Tying up Nicotine: New Selective Competitive Antagonist of the Neuronal Nicotinic Acetylcholine Receptors

Por Petersen, Ida Nymann, Crestey, François, Jensen, Anders A., Indurthi, Dinesh C., Pedersen, Henrik, Andreasen, Jesper T., Balle, Thomas, Kristensen, Jesper L.
Publicado no ACS Med Chem Lett (2015)

N-Hydroxypyrazolyl glycine derivatives as selective N-methyl-D-aspartic acid receptor ligands

Por Clausen, Rasmus P., Christensen, Caspar, Hansen, Kasper B., Greenwood, Jeremy R., Jørgensen, Lars, Micale, Nicola, Madsen, Jens Christian, Nielsen, Birgitte, Egebjerg, Jan, Bräuner-Osborne, Hans, Traynelis, Stephen F., Kristensen, Jesper L.
Publicado no J Med Chem (2008)

Serotonin 2A receptor agonist binding in the human brain with [(11)C]Cimbi-36

Por Ettrup, Anders, da Cunha-Bang, Sophie, McMahon, Brenda, Lehel, Szabolcs, Dyssegaard, Agnete, Skibsted, Anine W, Jørgensen, Louise M, Hansen, Martin, Baandrup, Anders O, Bache, Søren, Svarer, Claus, Kristensen, Jesper L, Gillings, Nic, Madsen, Jacob, Knudsen, Gitte M
Publicado em 2014