Synthesis and Evaluation of Dimeric Derivatives of Diacylglycerol–Lactones as Protein Kinase C Ligands

Autor Ohashi, Nami, Kobayashi, Ryosuke, Nomura, Wataru, Kobayakawa, Takuya, Czikora, Agnes, Herold, Brienna K., Lewin, Nancy E., Blumberg, Peter M., Tamamura, Hirokazu
Vydáno v Bioconjug Chem (2017)

Novel Radiolabeled Vanilloid with Enhanced Specificity for Human Transient Receptor Potential Vanilloid 1 (TRPV1)

Autor Pearce, Larry V., Ann, Jihyae, Jung, Aeran, Thorat, Shivaji A., Herold, Brienna K. A., Habtemichael, Amelework D., Blumberg, Peter M., Lee, Jeewoo
Vydáno v J Med Chem (2017)

Multi-Functional Diarylurea Small Molecule Inhibitors of TRPV1 with Therapeutic Potential for Neuroinflammation

Autor Feng, Zhiwei, Pearce, Larry V., Zhang, Yu, Xing, Changrui, Herold, Brienna K. A., Ma, Shifan, Hu, Ziheng, Turcios, Noe A., Yang, Peng, Tong, Qin, McCall, Anna K., Blumberg, Peter M., Xie, Xiang-Qun
Vydáno v AAPS J (2016)

Discovery of N-(3-fluoro-4-methylsulfonamidomethylphenyl)urea as a potent TRPV1 antagonistic template

Autor Ann, Jihyae, Sun, Wei, Zhou, Xing, Jung, Aeran, Baek, Jisoo, Lee, Sunho, Kim, Changhoon, Yoon, Suyoung, Hong, Sunhye, Choi, Sun, Turcios, Noe A., Herold, Brienna K. A., Esch, Timothy E., Lewin, Nancy E., Abramovitz, Adelle, Pearce, Larry V., Blumberg, Peter M., Lee, Jeewoo
Vydáno v Bioorg Med Chem Lett (2016)

2-Sulfonamidopyridine C-region analogs of 2-(3-fluoro-4-methylsulfonamidophenyl)propanamides as potent TRPV1 antagonists

Autor Ann, Jihyae, Ki, Yooran, Yoon, Suyoung, Kim, Myeong Seop, Lee, Jung-Un, Kim, Changhoon, Lee, Sunho, Jung, Aeran, Baek, Jisoo, Hong, Sunhye, Choi, Sun, Pearce, Larry V., Esch, Timothy E., Turcios, Noe A., Lewin, Nancy E., Ogunjirin, Adebowale E., Herold, Brienna K. A., McCall, Anna K., Blumberg, Peter M., Lee, Jeewoo
Vydáno v Bioorg Med Chem (2016)