Linear Free Energy Relationship Analysis of a Catalytic Desymmetrization Reaction of a Diarylmethane-Bis(phenol)

Por Gustafson, Jeffrey L., Sigman, Matthew S., Miller, Scott J.
Publicado em 2010

Dynamic Kinetic Resolution of Biaryl Atropisomers via Peptide-Catalyzed Asymmetric Bromination

Por Gustafson, Jeffrey L., Lim, Daniel, Miller, Scott J.
Publicado em 2010

Synthesis of Atropisomerically Defined, Highly Substituted Biaryl Scaffolds through Catalytic Enantioselective Bromination and Regioselective Cross-Coupling

Por Gustafson, Jeffrey L., Lim, Daniel, Barrett, Kimberly T., Miller, Scott J.
Publicado em 2011

A Case of Remote Asymmetric Induction in the Peptide-Catalyzed Desymmetrization of a Bis(phenol)

Por Lewis, Chad A., Gustafson, Jeffrey L., Chiu, Anna, Balsells, Jaume, Pollard, David, Murry, Jerry, Reamer, Robert A., Hansen, Karl B., Miller, Scott J.
Publicado em 2008

Identification of Hydrophobic Tags for the Degradation of Stabilized Proteins

Por Tae, Hyun Seop, Sundberg, Thomas B., Neklesa, Taavi K., Noblin, Devin J., Gustafson, Jeffrey L., Roth, Anke G., Raina, Kanak, Crews, Craig M.
Publicado em 2012

HaloPROTACS: Use of Small Molecule PROTACs to Induce Degradation of HaloTag Fusion Proteins

Por Buckley, Dennis L, Raina, Kanak, Darricarrere, Nicole, Hines, John, Gustafson, Jeffrey L, Smith, Ian E., Miah, Afjal H, Harling, John D, Crews, Craig M
Publicado no ACS Chem Biol (2015)

Small Molecule Inhibitors of the Interaction Between the E3 Ligase VHL and HIF1α

Por Buckley, Dennis L., Gustafson, Jeffrey L., Van Molle, Inge, Roth, Anke G., Tae, Hyun Seop, Gareiss, Peter C., Jorgensen, William L., Ciulli, Alessio, Crews, Craig M.
Publicado em 2012

Small Molecule Mediated Degradation of the Androgen Receptor Through Hydrophobic Tagging

Por Gustafson, Jeffrey L., Neklesa, Taavi K., Cox, Carly S., Roth, Anke G., Buckley, Dennis L., Tae, Hyun Seop, Sundberg, Thomas B., Stagg, D. Blake, Hines, John, McDonnell, Donald P., Norris, John D., Crews, Craig M.
Publicado no Angew Chem Int Ed Engl (2015)

Catalytic in vivo protein knockdown by small-molecule PROTACs

Por Bondeson, Daniel P, Mares, Alina, Smith, Ian E D, Ko, Eunhwa, Campos, Sebastien, Miah, Afjal H, Mulholland, Katie E, Routly, Natasha, Buckley, Dennis L, Gustafson, Jeffrey L, Zinn, Nico, Grandi, Paola, Shimamura, Satoko, Bergamini, Giovanna, Faelth-Savitski, Maria, Bantscheff, Marcus, Cox, Carly, Gordon, Deborah A, Willard, Ryan R, Flanagan, John J, Casillas, Linda N, Votta, Bartholomew J, den Besten, Willem, Famm, Kristoffer, Kruidenier, Laurens, Carter, Paul S, Harling, John D, Churcher, Ian, Crews, Craig M
Publicado no Nat Chem Biol (2015)