The G protein-coupled receptor subset of the rat genome

Por Gloriam, David E, Fredriksson, Robert, Schiöth, Helgi B
Publicado em 2007

SMARTCyp: A 2D Method for Prediction of Cytochrome P450-Mediated Drug Metabolism

Por Rydberg, Patrik, Gloriam, David E., Zaretzki, Jed, Breneman, Curt, Olsen, Lars
Publicado em 2010

The G protein-coupled receptor subset of the dog genome is more similar to that in humans than rodents

Por Haitina, Tatjana, Fredriksson, Robert, Foord, Steven M, Schiöth, Helgi B, Gloriam, David E
Publicado em 2009

Structure-Activity Relationships of Constrained Phenylethylamine Ligands for the Serotonin 5-HT(2) Receptors

Por Isberg, Vignir, Paine, James, Leth-Petersen, Sebastian, Kristensen, Jesper L., Gloriam, David E.
Publicado em 2013

Correction: Structure-Activity Relationships of Constrained Phenylethylamine Ligands for the Serotonin 5-HT(2) Receptors

Por Isberg, Vignir, Paine, James, Leth-Petersen, Sebastian, Kristensen, Jesper L., Gloriam, David E.
Publicado em 2014

Structural insight to mutation effects uncover a common allosteric site in class C GPCRs

Por Harpsøe, Kasper, Boesgaard, Michael W, Munk, Christian, Bräuner-Osborne, Hans, Gloriam, David E
Publicado no Bioinformatics (2017)

The G Protein–Coupled Receptor Subset of the Chicken Genome

Por Lagerström, Malin C, Hellström, Anders R, Gloriam, David E, Larsson, Thomas P, Schiöth, Helgi B, Fredriksson, Robert
Publicado em 2006

Pharmacogenomics of GPCR Drug Targets

Por Hauser, Alexander S., Chavali, Sreenivas, Masuho, Ikuo, Jahn, Leonie J., Martemyanov, Kirill A., Gloriam, David E., Babu, M. Madan
Publicado no Cell (2018)

Selective Negative Allosteric Modulation Of Metabotropic Glutamate Receptors – A Structural Perspective of Ligands and Mutants

Por Harpsøe, Kasper, Isberg, Vignir, Tehan, Benjamin G., Weiss, Dahlia, Arsova, Angela, Marshall, Fiona H., Bräuner-Osborne, Hans, Gloriam, David E.
Publicado no Sci Rep (2015)

Identification of Histamine H(3) Receptor Ligands Using a New Crystal Structure Fragment-based Method

Por Frandsen, Ida Osborn, Boesgaard, Michael W., Fidom, Kimberley, Hauser, Alexander S., Isberg, Vignir, Bräuner-Osborne, Hans, Wellendorph, Petrine, Gloriam, David E.
Publicado no Sci Rep (2017)

GPCRdb in 2018: adding GPCR structure models and ligands

Por Pándy-Szekeres, Gáspár, Munk, Christian, Tsonkov, Tsonko M, Mordalski, Stefan, Harpsøe, Kasper, Hauser, Alexander S, Bojarski, Andrzej J, Gloriam, David E
Publicado no Nucleic Acids Res (2018)

GPCRdb: an information system for G protein-coupled receptors

Por Isberg, Vignir, Mordalski, Stefan, Munk, Christian, Rataj, Krzysztof, Harpsøe, Kasper, Hauser, Alexander S., Vroling, Bas, Bojarski, Andrzej J., Vriend, Gert, Gloriam, David E.
Publicado no Nucleic Acids Res (2016)

GPCRdb: an information system for G protein-coupled receptors

Por Isberg, Vignir, Mordalski, Stefan, Munk, Christian, Rataj, Krzysztof, Harpsøe, Kasper, Hauser, Alexander S., Vroling, Bas, Bojarski, Andrzej J., Vriend, Gert, Gloriam, David E.
Publicado no Nucleic Acids Res (2017)

Novel Agonist Bioisosteres and Common Structure-Activity Relationships for The Orphan G Protein-Coupled Receptor GPR139

Por Shehata, Mohamed A., Nøhr, Anne C., Lissa, Delphine, Bisig, Christoph, Isberg, Vignir, Andersen, Kirsten B., Harpsøe, Kasper, Björkling, Fredrik, Bräuner-Osborne, Hans, Gloriam, David E.
Publicado no Sci Rep (2016)

Total synthesis and structure–activity relationship studies of a series of selective G protein inhibitors

Por Xiong, Xiao-Feng, Zhang, Hang, Underwood, Christina R., Harpsøe, Kasper, Gardella, Thomas J., Wöldike, Mie F., Mannstadt, Michael, Gloriam, David E., Bräuner-Osborne, Hans, Strømgaard, Kristian
Publicado no Nat Chem (2016)

Generic GPCR Residue Numbers - Aligning Topology Maps Minding The Gaps

Por Isberg, Vignir, de Graaf, Chris, Bortolato, Andrea, Cherezov, Vadim, Katritch, Vsevolod, Marshall, Fiona H., Mordalski, Stefan, Pin, Jean-Philippe, Stevens, Raymond C., Vriend, Gerrit, Gloriam, David E.
Publicado no Trends Pharmacol Sci (2014)

The orphan G protein-coupled receptor GPR139 is activated by the peptides: Adrenocorticotropic hormone (ACTH), α-, and β-melanocyte stimulating hormone (α-MSH, and β-MSH), and the...

Por Nøhr, Anne Cathrine, Shehata, Mohamed A., Hauser, Alexander S., Isberg, Vignir, Mokrosinski, Jacek, Andersen, Kirsten B., Farooqi, I. Sadaf, Pedersen, Daniel Sejer, Gloriam, David E., Bräuner-Osborne, Hans
Publicado no Neurochem Int (2017)

The GPR139 reference agonists 1a and 7c, and tryptophan and phenylalanine share a common binding site

Por Nøhr, Anne Cathrine, Jespers, Willem, Shehata, Mohamed A., Floryan, Leonard, Isberg, Vignir, Andersen, Kirsten Bayer, Åqvist, Johan, Gutiérrez-de-Terán, Hugo, Bräuner-Osborne, Hans, Gloriam, David E.
Publicado no Sci Rep (2017)

Development of a human vasopressin V(1a)-receptor antagonist from an evolutionary-related insect neuropeptide

Por Di Giglio, Maria Giulia, Muttenthaler, Markus, Harpsøe, Kasper, Liutkeviciute, Zita, Keov, Peter, Eder, Thomas, Rattei, Thomas, Arrowsmith, Sarah, Wray, Susan, Marek, Ales, Elbert, Tomas, Alewood, Paul F., Gloriam, David E., Gruber, Christian W.
Publicado no Sci Rep (2017)

A Community Standard Format for the Representation of Protein Affinity Reagents

Por Gloriam, David E., Orchard, Sandra, Bertinetti, Daniela, Björling, Erik, Bongcam-Rudloff, Erik, Borrebaeck, Carl A. K., Bourbeillon, Julie, Bradbury, Andrew R. M., de Daruvar, Antoine, Dübel, Stefan, Frank, Ronald, Gibson, Toby J., Gold, Larry, Haslam, Niall, Herberg, Friedrich W., Hiltke, Tara, Hoheisel, Jörg D., Kerrien, Samuel, Koegl, Manfred, Konthur, Zoltán, Korn, Bernhard, Landegren, Ulf, Montecchi-Palazzi, Luisa, Palcy, Sandrine, Rodriguez, Henry, Schweinsberg, Sonja, Sievert, Volker, Stoevesandt, Oda, Taussig, Michael J., Ueffing, Marius, Uhlén, Mathias, van der Maarel, Silvère, Wingren, Christer, Woollard, Peter, Sherman, David J., Hermjakob, Henning
Publicado em 2010