Stereoselective Inhibition of the hERG1 Potassium Channel

Por Grilo, Liliana Sintra, Carrupt, Pierre-Alain, Abriel, Hugues
Publicado em 2010

Quantitative structure-permeation relationship for iontophoretic transport across the skin

Por Mudry, Blaise, Carrupt, Pierre-Alain, Guy, Richard H., Delgado-Charro, M. Begoña
Publicado em 2007

Monoamine oxidase inhibitory properties of some benzazoles: Structure-; Activity relationships

Por Grandi, Teresa, Sparatore, Fabio, Gnerre, Carmela, Crivori, Patrizia, Carrupt, Pierre-Alain, Testa, Bernard
Publicado em 1999

HDAC6 as a target for neurodegenerative diseases: what makes it different from the other HDACs?

Por Simões-Pires, Claudia, Zwick, Vincent, Nurisso, Alessandra, Schenker, Esther, Carrupt, Pierre-Alain, Cuendet, Muriel
Publicado em 2013

Evidence for the existence of [(3)H]-trimetazidine binding sites involved in the regulation of the mitochondrial permeability transition pore

Por Morin, Didier, Elimadi, Aziz, Sapena, Rosa, Crevat, Aimé, Carrupt, Pierre-Alain, Testa, Bernard, Tillement, Jean-Paul
Publicado em 1998

Pharmacokinetics of β-adrenoceptor blockers in obese and normal volunteers

Por Cheymol, Georges, Poirier, Jean-Marie, Carrupt, Pierre-Alain, Testa, Bernard, Weissenburger, Jacques, Levron, Jean-Claude, Snoeck, Eric
Publicado em 1997

Entacapone and Tolcapone, Two Catechol O-Methyltransferase Inhibitors, Block Fibril Formation of α-Synuclein and β-Amyloid and Protect against Amyloid-induced Toxicity

Por Di Giovanni, Saviana, Eleuteri, Simona, Paleologou, Katerina E., Yin, Guowei, Zweckstetter, Markus, Carrupt, Pierre-Alain, Lashuel, Hilal A.
Publicado em 2010

Pharmacophore‐based discovery of inhibitors of a novel drug/proton antiporter in human brain endothelial hCMEC/D3 cell line

Por Chapy, Hélène, Goracci, Laura, Vayer, Philippe, Parmentier, Yannick, Carrupt, Pierre‐Alain, Declèves, Xavier, Scherrmann, Jean‐Michel, Cisternino, Salvatore, Cruciani, Gabriele
Publicado no Br J Pharmacol (2015)

A Rational Approach for the Identification of Non-Hydroxamate HDAC6-Selective Inhibitors

Por Goracci, Laura, Deschamps, Nathalie, Randazzo, Giuseppe Marco, Petit, Charlotte, Dos Santos Passos, Carolina, Carrupt, Pierre-Alain, Simões-Pires, Claudia, Nurisso, Alessandra
Publicado no Sci Rep (2016)

Computational Studies on Sirtuins from Trypanosoma cruzi: Structures, Conformations and Interactions with Phytochemicals

Por Sacconnay, Lionel, Angleviel, Melissa, Randazzo, Giuseppe Marco, Marçal Ferreira Queiroz, Marcos, Ferreira Queiroz, Emerson, Wolfender, Jean-Luc, Carrupt, Pierre-Alain, Nurisso, Alessandra
Publicado em 2014