Resultados da pesquisa - ((((((((eur j) OR (mur j))) OR (eus j))) OR (kur j))) OR (((eun a) OR (sun j)))) med chem

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Editorial – IChemE Special Issue on Climate Change

Por Pritchard, EurIng Colin
Publicado no Chem Eng Res Des (2020)

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(S)-4-Trimethylsilyl-3-butyn-2-ol as an auxiliary for stereocontrolled synthesis of salinosporamide analogs with modifications at positions C2 and C5

Por Blasdel, Landy K., Lee, DongEun, Sun, Binyuan, Myers, Andrew G.
Publicado em 2013

“...Analogs of salinsporamide A with variations of the C2 and C5 substituents are prepared in 8–10...”
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Reprofiling of pyrimidine-based DAPK1/CSF1R dual inhibitors: identification of 2,5-diamino-4-pyrimidinol derivatives as novel potential anticancer lead compounds

Por Farag, Ahmed K., Hassan, Ahmed H. E., Ahn, Byung Sun, Park, Ki Duk, Roh, Eun Joo
Publicado no J Enzyme Inhib Med Chem (2019)

“... with 2-anilino-4-phenoxypyrimidines suggests a series of 2,5-diamino-4-pyrimidinol derivatives...”
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The carbonate analogues of 5′-halogenated resiniferatoxin as TRPV1 ligands

Por Lim, Kwang Su, Lee, Hobin, Kim, Sung Eun, Ha, Tae-Hwan, Ann, Jihyae, Son, Karam, Choi, Sun, Sun, Wei, Pearce, Larry V., DeAndrea-Lazarus, Ian A., Blumberg, Peter M., Lee, Jeewoo
Publicado no Eur J Med Chem (2013)

“...A series of carbonate analogues of 5′-halogenated RTX have been investigated in order to examine...”
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Structure-activity relationships and docking studies of synthetic 2-arylindole derivatives determined with aromatase and quinone reductase 1

Por Prior, Allan M., Yu, Xufen, Park, Eun-Jung, Kondratyuk, Tamara P., Lin, Yan, Pezzuto, John M., Sun, Dianqing
Publicado no Bioorg Med Chem Lett (2017)

“...In our ongoing effort of discovering anticancer and chemopreventive agents, a series of 2...”
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Design, synthesis, and biological evaluation of callophycin A and analogues as potential chemopreventive and anticancer agents

Por Shen, Li, Park, Eun-Jung, Kondratyuk, Tamara P., Guendisch, Daniela, Marler, Laura, Pezzuto, John M., Wright, Anthony D., Sun, Dianqing
Publicado em 2011

“...Callophycin A was originally isolated from the red algae Callophycus oppositifolius and shown...”
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Structure–Activity Studies of Divin: An Inhibitor of Bacterial Cell Division

Por Zhou, Maoquan, Eun, Ye-Jin, Guzei, Ilia A., Weibel, Douglas B.
Publicado em 2013

“... of divin, a small molecule that blocks bacterial division by perturbing the assembly of proteins...”
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Asymmetric synthesis and receptor activity of chiral simplified resiniferatoxin (sRTX) analogues as transient receptor potential vanilloid 1 (TRPV1) ligands

Por Kim, Myeong Seop, Ki, Yooran, Ahn, Song Yeon, Yoon, Suyoung, Kim, Sung-Eun, Park, Hyeung-Geun, Sun, Wei, Son, Karam, Cui, Minghua, Choi, Sun, Pearce, Larry V., Esch, Timothy E., DeAndrea-Lazarus, Ian A., Blumberg, Peter M., Lee, Jeewoo
Publicado no Bioorg Med Chem Lett (2013)

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Cyclic opioid peptides

Por Remesic, Michael, Lee, Yeon Sun, Hruby, Victor J.
Publicado no Curr Med Chem (2016)

“... of pain. Since the first discovery of enkephalin, approximately a dozen endogenous opioid peptides have...”
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Simultaneous determination of methylcarbamate and ethylcarbamate in fermented foods and beverages by derivatization and GC-MS analysis

Por Shin, Ho-Sang, Yang, Eun-Young
Publicado em 2012

“... in fermented food and beverages. In order to estimate the risk for their exposure, a sensitive simultaneous...”
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Synthesis and evaluation of bivalent ligands for binding to the human melanocortin-4 receptor

Por Fernandes, Steve M., Lee, Yeon Sun, Gillies, Robert J., Hruby, Victor J.
Publicado no Bioorg Med Chem (2014)

“..., synthesized, and tested a series of bivalent ligands targeting the over-expressed human melanocortin 4...”
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Structure Activity Relationships of 1,4-Dihydropyridines That Act as Enhancers of the Vanilloid Receptor 1 (TRPV1)

Por Roh, Eun Joo, Keller, Jason M., Olah, Zoltan, Iadarola, Michael J., Jacobson, Kenneth A.
Publicado em 2008

“...Vanilloid agonists such as capsaicin activate ion flux through the TRPV1 channel, a heat...”
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Dynorphin A analogs for the treatment of chronic neuropathic pain

Por Hall, Sara M, Lee, Yeon Sun, Hruby, Victor J
Publicado no Future Med Chem (2016)

“... states. The endogenous peptide, dynorphin A has long been established as a target for the treatment...”
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CRISPR/dCas9-mediated biosensor for detection of tick-borne diseases

Por Koo, Bonhan, Kim, Da-eun, Kweon, Jiyeon, Jin, Choong Eun, Kim, Sung-Han, Kim, Yongsub, Shin, Yong
Publicado no Sens Actuators B Chem (2018)

“... tool that utilizes CRISPR/dCas9-mediated biosensor that couples a nuclease inactivated Cas9 (dCas9...”
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Pathogenic Bacterial Proteins and their Anti-Inflammatory Effects in the Eukaryotic Host

Por Sun, Jun
Publicado em 2009

“... Salmonella AvrA, Enteropathogenic Escherichia coli Cif, and Yersinia YopJ, Staphylococcus aureus...”
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Redefining the structure-activity relationships of 2,6-methano-3-benzazocines. 6. Opioid receptor binding properties of cyclic variants of 8-carboxamidocyclazocine

Por Wentland, Mark P., Sun, Xufeng, Cohen, Dana J., Bidlack, Jean M.
Publicado em 2008

“...A series of 7,8- and 8,9-fused pyrimidinone, aminopyridine and pyridone derivatives of 8...”
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Small molecule inhibitors in pancreatic cancer

Por Sun, Jufeng, Russell, Cecilia C., Scarlett, Christopher J., McCluskey, Adam
Publicado no RSC Med Chem (2020)

“...Pancreatic cancer (PC), with a 5 year survival of <7%, is one of the most fatal of all human...”
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Design and synthesis of de novo cytotoxic alkaloids by mimicking the bioactive conformation of paclitaxel

Por Sun, Liang, Veith, Jean M., Pera, Paula, Bernacki, Ralph J., Ojima, Iwao
Publicado em 2010

“...Novel paclitaxel-mimicking alkaloids were designed and synthesized based on a bioactive...”
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2-(3-Fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists: Structure activity relationships of the 2-oxy pyridine C-region

Por Thorat, Shivaji A., Kang, Dong Wook, Ryu, HyungChul, Kim, Myeong Seop, Kim, Ho Shin, Ann, Jihyae, Ha, Taehwan, Kim, Sung-Eun, Son, Karam, Choi, Sun, Blumberg, Peter M., Frank, Robert, Bahrenberg, Gregor, Schiene, Klaus, Christoph, Thomas, Lee, Jeewoo
Publicado no Eur J Med Chem (2013)

“... analysis of 53S using our hTRPVl homology model indicated that the A- and B-region 2-(3-fluoro-4...”
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Synthesis and Biological Evaluation of Manassantin Analogues for Hypoxia-Inducible Factor 1α Inhibition

Por Kwon, Do-Yeon, Lee, Hye Eun, Weitzel, Douglas H., Park, Kyunghye, Lee, Sun Hee, Lee, Chen-Ting, Stephenson, Tesia N., Park, Hyeri, Fitzgerald, Michael C., Chi, Jen-Tsan, Mook, Robert A., Dewhirst, Mark W., Lee, You Mie, Hong, Jiyong
Publicado no J Med Chem (2015)

“...[Image: see text] To cope with hypoxia, tumor cells have developed a number of adaptive mechanisms...”
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