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Targeting Protein Kinases Degradation by PROTACs

Kinase dysregulation is greatly associated with cell proliferation, migration and survival, indicating the importance of kinases as therapeutic targets for anticancer drug development. However, traditional kinase inhibitors binding to catalytic or allosteric sites are associated with significant cha...

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Bibliografski detalji
Izdano u:Front Chem
Glavni autori: Yu, Fei, Cai, Ming, Shao, Liang, Zhang, Jihong
Format: Artigo
Jezik:Inglês
Izdano: Frontiers Media S.A. 2021
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC8279777/
https://ncbi.nlm.nih.gov/pubmed/34277564
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fchem.2021.679120
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