Laddar...

Homotropic Cooperativity of Midazolam Metabolism by Cytochrome P450 3A4: Insight from Computational Studies

[Image: see text] Human cytochrome P450 3A4 (CYP3A4) is responsible for the metabolism of ∼50% clinically used drugs. Midazolam (MDZ) is a commonly used sedative drug and serves as a marker substrate for the CYP3A4 activity assessment. MDZ is metabolized by CYP3A4 to two hydroxylation products, 1′-O...

Full beskrivning

Sparad:
Bibliografiska uppgifter
I publikationen:J Chem Inf Model
Huvudupphovsmän: Li, Junhao, Chen, Yue, Tang, Yun, Li, Weihua, Tu, Yaoquan
Materialtyp: Artigo
Språk:Inglês
Publicerad: American Chemical Society 2021
Länkar:https://ncbi.nlm.nih.gov/pmc/articles/PMC8278384/
https://ncbi.nlm.nih.gov/pubmed/33884878
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jcim.1c00266
Taggar: Lägg till en tagg
Inga taggar, Lägg till första taggen!