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Multi-Target Directed Ligands (MTDLs) Binding the σ(1) Receptor as Promising Therapeutics: State of the Art and Perspectives

The sigma-1 (σ(1)) receptor is a ‘pluripotent chaperone’ protein mainly expressed at the mitochondria–endoplasmic reticulum membrane interfaces where it interacts with several client proteins. This feature renders the σ(1) receptor an ideal target for the development of multifunctional ligands, whos...

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Dettagli Bibliografici
Pubblicato in:Int J Mol Sci
Autori principali: Abatematteo, Francesca Serena, Niso, Mauro, Contino, Marialessandra, Leopoldo, Marcello, Abate, Carmen
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2021
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC8232171/
https://ncbi.nlm.nih.gov/pubmed/34198620
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms22126359
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