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Drugging the Undruggable: Advances on RAS Targeting in Cancer

Around 20% of all malignancies harbour activating mutations in RAS isoforms. Despite this, there is a deficiency of RAS-targeting agents licensed for therapeutic use. The picomolar affinity of RAS for GTP, and the lack of suitable pockets for high-affinity small-molecule binding, precluded effective...

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書目詳細資料
發表在:Genes (Basel)
Main Authors: Molina-Arcas, Miriam, Samani, Amit, Downward, Julian
格式: Artigo
語言:Inglês
出版: MDPI 2021
主題:
在線閱讀:https://ncbi.nlm.nih.gov/pmc/articles/PMC8228461/
https://ncbi.nlm.nih.gov/pubmed/34200676
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/genes12060899
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