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Discovery of a Small Side Cavity in Sphingosine Kinase 2 that Enhances Inhibitor Potency and Selectivity

The sphingosine-1-phosphate (S1P) signaling pathway is an attractive drug target due to its involvement in immune cell chemotaxis and vascular integrity. The formation of S1P is catalyzed by sphingosine kinase 1 or 2 (SphK1 or SphK2) from sphingosine (Sph) and ATP. Inhibition of SphK1 and 2 to atten...

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Detalhes bibliográficos
Publicado no:J Med Chem
Main Authors: Sibley, Christopher D., Morris, Emily A., Kharel, Yugesh, Brown, Anne M., Bevan, David R., Lynch, Kevin R., Santos, Webster L.
Formato: Artigo
Idioma:Inglês
Publicado em: 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC8215855/
https://ncbi.nlm.nih.gov/pubmed/31895563
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.9b01508
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