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Mining for METTL3 inhibitors to suppress cancer

The RNA methyltransferase METTL3 catalyzes N(6)-methyladenosine (m(6)A) modification of messenger RNAs (mRNAs). It is overexpressed in many types of cancer, including acute myelogenous leukemia (AML), and promotes cancer cell growth and tumorigenicity. Now, a selective small molecule inhibitor of ME...

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Detalles Bibliográficos
Publicado en:Nat Struct Mol Biol
Main Authors: Li, Jiazhi, Gregory, Richard I.
Formato: Artigo
Idioma:Inglês
Publicado: 2021
Assuntos:
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC8197751/
https://ncbi.nlm.nih.gov/pubmed/34040230
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41594-021-00606-5
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