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Alterations in the global proteome and phosphoproteome in third-generation EGFR TKI resistance reveal drug targets to circumvent resistance

Lung cancer is the leading cause of cancer mortality worldwide. The treatment of lung cancer patients harboring mutant EGFR with orally administered EGFR tyrosine kinase inhibitors (TKIs) has been a paradigm shift. Osimertinib and rociletinib are third-generation irreversible EGFR TKIs targeting the...

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Dettagli Bibliografici
Pubblicato in:Cancer Res
Autori principali: Zhang, Xu, Maity, Tapan K., Ross, Karen E., Qi, Yue, Cultraro, Constance M., Bahta, Meriam, Pitts, Stephanie, Keswani, Meghana, Gao, Shaojian, Nguyen, Khoa Dang P., Cowart, Julie, Kirkali, Fatos, Wu, Cathy, Guha, Udayan
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2021
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC8182571/
https://ncbi.nlm.nih.gov/pubmed/33727228
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/0008-5472.CAN-20-2435
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