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α-Methylene-β-Lactone Scaffold for Developing Chemical Probes at the Two Ends of the Selectivity Spectrum

The utilities of an α-methylene-β-lactone (MeLac) moiety as a warhead composed of multiple electrophilic sites are reported. We demonstrate that a MeLac-alkyne not only reacts with diverse proteins as a broadly reactive measurement probe but also recruits reduced endogenous glutathione (GSH) to asse...

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Bibliografische gegevens
Gepubliceerd in:Chembiochem
Hoofdauteurs: Wang, Lei, Riel, Louis P., Bajrami, Bekim, Deng, Bin, Howell, Amy R., Yao, Xudong
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: 2020
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Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC8114233/
https://ncbi.nlm.nih.gov/pubmed/32964640
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cbic.202000605
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