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Allosterism vs. Orthosterism: Recent Findings and Future Perspectives on A(2B) AR Physio-Pathological Implications

The development of GPCR (G-coupled protein receptor) allosteric modulators has attracted increasing interest in the last decades. The use of allosteric modulators in therapy offers several advantages with respect to orthosteric ones, as they can fine-tune the tissue responses to the endogenous agoni...

Täydet tiedot

Tallennettuna:
Bibliografiset tiedot
Julkaisussa:Front Pharmacol
Päätekijät: Barresi, Elisabetta, Martini, Claudia, Da Settimo, Federico, Greco, Giovanni, Taliani, Sabrina, Giacomelli, Chiara, Trincavelli, Maria Letizia
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: Frontiers Media S.A. 2021
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC8024542/
https://ncbi.nlm.nih.gov/pubmed/33841166
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fphar.2021.652121
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