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TSPO PIGA Ligands Promote Neurosteroidogenesis and Human Astrocyte Well-Being

The steroidogenic 18 kDa translocator protein (TSPO) is an emerging, attractive therapeutic tool for several pathological conditions of the nervous system. Here, 13 high affinity TSPO ligands belonging to our previously described N,N-dialkyl-2-phenylindol-3-ylglyoxylamide (PIGA) class were evaluated...

Полное описание

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Библиографические подробности
Опубликовано в: :Int J Mol Sci
Главные авторы: Da Pozzo, Eleonora, Giacomelli, Chiara, Costa, Barbara, Cavallini, Chiara, Taliani, Sabrina, Barresi, Elisabetta, Da Settimo, Federico, Martini, Claudia
Формат: Artigo
Язык:Inglês
Опубликовано: MDPI 2016
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC4964404/
https://ncbi.nlm.nih.gov/pubmed/27367681
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms17071028
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