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TSPO PIGA Ligands Promote Neurosteroidogenesis and Human Astrocyte Well-Being

The steroidogenic 18 kDa translocator protein (TSPO) is an emerging, attractive therapeutic tool for several pathological conditions of the nervous system. Here, 13 high affinity TSPO ligands belonging to our previously described N,N-dialkyl-2-phenylindol-3-ylglyoxylamide (PIGA) class were evaluated...

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Detalles Bibliográficos
Publicado en:Int J Mol Sci
Main Authors: Da Pozzo, Eleonora, Giacomelli, Chiara, Costa, Barbara, Cavallini, Chiara, Taliani, Sabrina, Barresi, Elisabetta, Da Settimo, Federico, Martini, Claudia
Formato: Artigo
Idioma:Inglês
Publicado: MDPI 2016
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4964404/
https://ncbi.nlm.nih.gov/pubmed/27367681
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms17071028
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