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Structure and selectivity engineering of the M(1) muscarinic receptor toxin complex

Muscarinic toxins (MTs) are natural toxins produced by mamba snakes that primarily bind to muscarinic acetylcholine receptors (MAChRs) and modulate their function. Despite their similar primary and tertiary structures, MTs show distinct binding selectivity toward different MAChRs. The molecular deta...

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Detalhes bibliográficos
Publicado no:Science
Main Authors: Maeda, Shoji, Xu, Jun, Kadji, Francois Marie N., Clark, Mary J., Zhao, Jiawei, Tsutsumi, Naotaka, Aoki, Junken, Sunahara, Roger K., Inoue, Asuka, Garcia, K Christopher, Kobilka, Brian K.
Formato: Artigo
Idioma:Inglês
Publicado em: 2020
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7954660/
https://ncbi.nlm.nih.gov/pubmed/32646996
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1126/science.aax2517
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