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Inhibition of HER Receptors Reveals Distinct Mechanisms of Compensatory Upregulation of Other HER Family Members: Basis for Acquired Resistance and for Combination Therapy

Overexpression of members of the HER/erbB transmembrane tyrosine kinase family like HER2/erbB2/neu is associated with various cancers. Some heterodimers, especially HER2/HER3 heterodimers, are particularly potent inducers of oncogenic signaling. Still, from a clinical viewpoint their inhibition has...

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Publicat a:Cells
Autors principals: Gutsch, Daniela, Jenke, Robert, Büch, Thomas, Aigner, Achim
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2021
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7911202/
https://ncbi.nlm.nih.gov/pubmed/33572976
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/cells10020272
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