Selective inhibition of carbonic anhydrase IX and XII by coumarin and psoralen derivatives

A small library of coumarin and their psoralen analogues EMAC10157a-b-d-g and EMAC10160a-b-d-g has been designed and synthesised to investigate the effect of structural modifications on their inhibition ability and selectivity profile towards carbonic anhydrase isoforms I, II, IX, and XII. None of t...

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Détails bibliographiques
Publié dans:J Enzyme Inhib Med Chem
Auteurs principaux: Meleddu, Rita, Deplano, Serenella, Maccioni, Elias, Ortuso, Francesco, Cottiglia, Filippo, Secci, Daniela, Onali, Alessia, Sanna, Erica, Angeli, Andrea, Angius, Rossella, Alcaro, Stefano, Supuran, Claudiu T., Distinto, Simona
Format: Artigo
Langue:Inglês
Publié: Taylor & Francis 2021
Sujets:
Brief Report
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC7899656/
https://ncbi.nlm.nih.gov/pubmed/33602041
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/14756366.2021.1887171
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