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Inhibition of Nonfunctional Ras

Intuitively, functional states should be targeted; not nonfunctional ones. So why could drugging the inactive K-Ras4B(G12C) work – but, drugging the inactive kinase will likely not? The reason is the distinct oncogenic mechanisms. Kinase driver mutations work by stabilizing the active state and/or d...

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Sonraí Bibleagrafaíochta
Foilsithe in:Cell Chem Biol
Main Authors: Nussinov, Ruth, Jang, Hyunbum, Gursoy, Attila, Keskin, Ozlem, Gaponenko, Vadim
Formáid: Artigo
Teanga:Inglês
Foilsithe: 2021
Ábhair:
Rochtain Ar Líne:https://ncbi.nlm.nih.gov/pmc/articles/PMC7897307/
https://ncbi.nlm.nih.gov/pubmed/33440168
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.chembiol.2020.12.012
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