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Building a Chemical Toolbox for Human Pregnane X Receptor Research: Discovery of Agonists, Inverse Agonists, and Antagonists Among Analogs based on the Unique Chemical Scaffold of SPA70
Pregnane X receptor (PXR) plays roles in detoxification and other physiologic processes. PXR activation may enhance drug metabolism (leading to adverse drug reactions) or inhibit inflammation. Therefore, PXR agonists, antagonists, and inverse agonists may serve as research tools and drug candidates....
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| Publicado en: | J Med Chem |
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| Autores principales: | , , , , , |
| Formato: | Artigo |
| Lenguaje: | Inglês |
| Publicado: |
2021
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| Materias: | |
| Acceso en línea: | https://ncbi.nlm.nih.gov/pmc/articles/PMC7880548/ https://ncbi.nlm.nih.gov/pubmed/33497575 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.0c02201 |
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