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Exploration of Structure–Activity Relationship of Aromatic Aldehydes Bearing Pyridinylmethoxy-Methyl Esters as Novel Antisickling Agents

Aromatic aldehydes elicit their antisickling effects primarily by increasing the affinity of hemoglobin (Hb) for oxygen (O(2)). However, challenges related to weak potency and poor pharmacokinetic properties have hampered their development to treat sickle cell disease (SCD). Herein, we report our ef...

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Detalhes bibliográficos
Publicado no:J Med Chem
Main Authors: Pagare, Piyusha P., Ghatge, Mohini S., Chen, Qiukan, Musayev, Faik N., Venitz, Jurgen, Abdulmalik, Osheiza, Zhang, Yan, Safo, Martin K.
Formato: Artigo
Idioma:Inglês
Publicado em: 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7869023/
https://ncbi.nlm.nih.gov/pubmed/33205981
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.0c01287
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