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Structure-Guided Computational Methods Predict Multiple Distinct Binding Modes for Pyrazoloquinolinones in GABA(A) Receptors

Pyrazoloquinolinones (PQs) are a versatile class of GABA(A) receptor ligands. It has been demonstrated that high functional selectivity for certain receptor subtypes can be obtained by specific substitution patterns, but so far, no clear SAR rules emerge from the studies. As is the case for many GAB...

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Detalhes bibliográficos
Publicado no:Front Neurosci
Main Authors: Fabjan, Jure, Koniuszewski, Filip, Schaar, Benjamin, Ernst, Margot
Formato: Artigo
Idioma:Inglês
Publicado em: Frontiers Media S.A. 2021
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7844064/
https://ncbi.nlm.nih.gov/pubmed/33519364
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fnins.2020.611953
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