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Cellular Uptake and Cytosolic Delivery of a Cyclic Cystine Knot Scaffold

Cyclotides are macrocyclic peptides with exceptionally stable structures and have been reported to penetrate cells, making them promising scaffolds for the delivery of inhibitory peptides to target intracellular proteins. However, their cellular uptake and cytosolic localization have been poorly und...

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Dettagli Bibliografici
Pubblicato in:ACS Chem Biol
Autori principali: Yin, Huawu, Huang, Yen-Hua, Deprey, Kirsten, Condon, Nicholas D., Kritzer, Joshua A., Craik, David J., Wang, Conan K.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7831380/
https://ncbi.nlm.nih.gov/pubmed/32315152
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschembio.0c00297
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