Loading...

Meloxicam methyl group determines enzyme specificity for thiazole bioactivation compared to sudoxicam

Meloxicam is a thiazole-containing NSAID that was approved for marketing with favorable clinical outcomes despite being structurally similar to the hepatotoxic sudoxicam. Introduction of a single methyl group on the thiazole results in an overall lower toxic risk, yet the group’s impact on P450 isoz...

Fuld beskrivelse

Na minha lista:
Bibliografiske detaljer
Udgivet i:Toxicol Lett
Main Authors: Barnette, Dustyn A., Schleiff, Mary A., Datta, Arghya, Flynn, Noah, Swamidass, S. Joshua, Miller, Grover P.
Format: Artigo
Sprog:Inglês
Udgivet: 2020
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC7807415/
https://ncbi.nlm.nih.gov/pubmed/33253783
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.toxlet.2020.11.015
Tags: Tilføj Tag
Ingen Tags, Vær først til at tagge denne postø!