Carregant...

Pharmacological Characterization of µ-Opioid Receptor Agonists with Biased G Protein or β-Arrestin Signaling, and Computational Study of Conformational Changes during Receptor Activation

In recent years, G protein vs. β-arrestin biased agonism at opioid receptors has been proposed as an opportunity to produce antinociception with reduced adverse effects. However, at present this approach is highly debated, a reason why more information about biased ligands is required. While the pra...

Descripció completa

Guardat en:
Dades bibliogràfiques
Publicat a:Molecules
Autors principals: Piekielna-Ciesielska, Justyna, Artali, Roberto, Azzam, Ammar A. H., Lambert, David G., Kluczyk, Alicja, Gentilucci, Luca, Janecka, Anna
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2020
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7792944/
https://ncbi.nlm.nih.gov/pubmed/33375124
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules26010013
Etiquetes: Afegir etiqueta
Sense etiquetes, Sigues el primer a etiquetar aquest registre!