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Identification of a New Heterocyclic Scaffold for Inhibitors of the Polo-Box Domain of Polo-like Kinase 1

As a mitotic-specific target widely deregulated in various human cancers, polo-like kinase 1 (Plk1) has been extensively explored for anticancer activity and drug discovery. Although multiple catalytic domain inhibitors were tested in preclinical and clinical studies, their efficacies are limited by...

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Publicado en:J Med Chem
Main Authors: Alverez, Celeste N., Park, Jung-Eun, Toti, Kiran S., Xia, Yangliu, Krausz, Kristopher W., Rai, Ganesha, Bang, Jeong K., Gonzalez, Frank J., Jacobson, Kenneth A., Lee, Kyung S.
Formato: Artigo
Idioma:Inglês
Publicado: 2020
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC7769008/
https://ncbi.nlm.nih.gov/pubmed/33175530
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.0c01669
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