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Enantiomer-specific activities of an LRH-1 and SF-1 dual agonist

Chirality is an important consideration in drug development: it can influence recognition of the intended target, pharmacokinetics, and off-target effects. Here, we investigate how chirality affects the activity and mechanism of action of RJW100, a racemic agonist of the nuclear receptors liver rece...

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Detalhes bibliográficos
Publicado no:Sci Rep
Main Authors: Mays, Suzanne G., Stec, Józef, Liu, Xu, D’Agostino, Emma H., Whitby, Richard J., Ortlund, Eric A.
Formato: Artigo
Idioma:Inglês
Publicado em: Nature Publishing Group UK 2020
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7747700/
https://ncbi.nlm.nih.gov/pubmed/33335203
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-020-79251-9
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