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Stability and cell permeability of sulfonyl fluorides in the design of Lys-covalent antagonists of protein-protein interactions

Recently we reported on aryl-fluorosulfates as possible stable and effective electrophiles for the design of lysine covalent, cell permeable antagonists of protein-protein interactions (PPIs). Here we revisit the use of aryl-sulfonyl fluorides as Lys-targeting moieties, incorporating these electroph...

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Vydáno v:ChemMedChem
Hlavní autoři: Gambini, Luca, Udompholkul, Parima, Salem, Ahmed F., Baggio, Carlo, Pellecchia, Maurizio
Médium: Artigo
Jazyk:Inglês
Vydáno: 2020
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7722097/
https://ncbi.nlm.nih.gov/pubmed/32790900
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cmdc.202000355
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